WNK inhibitor 7

CAS No. 2125724-72-1

WNK inhibitor 7( WNK-IN-7 | WNK IN 7 | WNKIN7 | WNK inhibitor 7 | WNK inhibitor-7 )

Catalog No. M13379 CAS No. 2125724-72-1

A potent, selectiive inhibitor of WNK1 kinase with IC50 of 95 nM, shows IC50 of 1.39 uM in the cellular OSR1 phosphorylation assay with reasonable aqueous solubility.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    WNK inhibitor 7
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent, selectiive inhibitor of WNK1 kinase with IC50 of 95 nM, shows IC50 of 1.39 uM in the cellular OSR1 phosphorylation assay with reasonable aqueous solubility.
  • Description
    A potent, selectiive inhibitor of WNK1 kinase with IC50 of 95 nM, shows IC50 of 1.39 uM in the cellular OSR1 phosphorylation assay with reasonable aqueous solubility.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    WNK-IN-7 | WNK IN 7 | WNKIN7 | WNK inhibitor 7 | WNK inhibitor-7
  • Pathway
    Autophagy
  • Target
    WNK Kinase
  • Recptor
    WNK Kinase
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2125724-72-1
  • Formula Weight
    399.538
  • Molecular Formula
    C26H29N3O
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CC(C)CNCC1=CN(C2=CC(C3=CC=CC(OC)=C3)=NC=C2C)C4=C1C=CC=C4
  • Chemical Name
    N-((1-(2-(3-methoxyphenyl)-5-methylpyridin-4-yl)-1H-indol-3-yl)methyl)-2-methylpropan-1-amine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Yamada K, et al. ACS Chem Biol. 2016 Dec 16;11(12):3338-3346.
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